SCHEMBL6446641

SCHEMBL6446641

N#CCNC(=O)C(CNC(=O)c1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.64
GPR139 Q6DWJ6 1/20 0.56
TACR1 P25103 1/20 0.54
ALDH1A1 P00352 2/20 0.52
POLB P06746 2/20 0.52
CTSK P43235 3/20 0.52
CTSS P25774 2/20 0.52
NPC1 O15118 1/20 0.49
MEN1 O00255 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.47
TP53BP1 Q12888 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822952 0.93 CTSL (0.61) CTSLGPR139TACR1ALDH1A1POLB
SCHEMBL6444047 0.91 CTSL (0.53) CTSLGPR139TACR1ALDH1A1POLB
SCHEMBL6446794 0.90 CTSL (0.58) CTSLGPR139TACR1ALDH1A1POLB
SCHEMBL5517758 0.85 CTSK (0.61) CTSLCTSKCTSSNPC1SMN1; SMN2
SCHEMBL6824499 0.83 CTSL (0.62) CTSLGPR139TACR1ALDH1A1POLB
SCHEMBL27457044 0.83 POLB (0.68) CTSLGPR139ALDH1A1POLBNPSR1
SCHEMBL6445446 0.83 CTSL (0.55) CTSLGPR139TACR1ALDH1A1POLB
SCHEMBL6446138 0.83 CTSL (0.61) CTSLGPR139ALDH1A1POLBNPC1
SCHEMBL6442129 0.83 CTSL (0.49) CTSLGPR139TACR1ALDH1A1POLB
SCHEMBL6447506 0.81 CTSL (0.53) CTSLCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed