SCHEMBL6447552

SCHEMBL6447552

N#CCNC(=O)C(CNC(=O)c1ccc(CCl)cc1)c1csc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.42
CTSL P07711 10/20 0.42
CTSS P25774 9/20 0.42
CTSB P07858 5/20 0.40
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448205 0.91 CTSL (0.47) CTSKCTSLCTSSCTSB
SCHEMBL6443534 0.91 HDAC6 (0.37) CTSKCTSLCTSSHDAC1HDAC6
SCHEMBL6446814 0.90 CTSL (0.41) CTSKCTSLCTSSCTSB
SCHEMBL6446486 0.86 CTSK (0.41) CTSKCTSLCTSSCTSBHDAC6
SCHEMBL6021296 0.82 CTSL (0.38) CTSKCTSLCTSSCTSBHDAC1
SCHEMBL6021888 0.82 CTSK (0.44) CTSKCTSLCTSSCTSBHDAC1
SCHEMBL6444782 0.81 CTSK (0.53) CTSKCTSLCTSSCTSB
SCHEMBL6446480 0.81 GUSB (0.36) CTSKCTSLCTSSCTSBHDAC6
SCHEMBL6443383 0.81 CTSS (0.51) CTSKCTSLCTSSCTSB
SCHEMBL6821937 0.80 CTSK (0.43) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed