SCHEMBL6441382

SCHEMBL6441382

CSc1ccc(-c2[nH]nc(CCCC(=O)O)c2-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
PPARG P37231 5/20 0.36
PPARD Q03181 5/20 0.36
PPARA Q07869 4/20 0.35
NR1H4 Q96RI1 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
GPR35 Q9HC97 1/20 0.35
FFAR1 O14842 1/20 0.34
EPHX2 P34913 1/20 0.34
LTB4R Q15722 2/20 0.34
MLYCD O95822 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
GSK3B P49841 2/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445697 0.84 PTGDR2 (0.44) NR1H4PTGDR2
SCHEMBL6444469 0.74 ALDH1A1 (0.41) POLBKDM4ENPC1RAB9AATM
SCHEMBL6440587 0.71 POLB (0.36) POLBKDM4ENPC1RAB9AATM
SCHEMBL6438861 0.70 RPS6KA3 (0.43) KDM4ENPC1RAB9AGSK3B
SCHEMBL3870144 0.69 RXRA (0.56) NR1H4EPHX2
SCHEMBL8637993 0.67 RXFP1 (0.34) POLBMAPTGSK3BMAPK14
SCHEMBL17077274 0.67 KIF11 (0.50) PPARGPPARDPPARAGSK3B
SCHEMBL46638 0.64 HSD17B10 (0.61) NR1H4MAPTFFAR1
SCHEMBL1454387 0.64 FFAR1 (0.60) PPARGPPARANR1H4MAPTFFAR1
SCHEMBL30741037 0.64 KDM4E (0.43) KDM4ENPC1RAB9AATMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed