SCHEMBL6448790

SCHEMBL6448790

CC(C)NC(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)NC(C)C

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60
LMNA P02545 1/20 0.49
CA2 P00918 1/20 0.46
NAALAD2 Q9Y3Q0 2/20 0.45
FOLH1 Q04609 1/20 0.45
TAAR1 Q96RJ0 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
CTRB1 P17538 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448962 0.81 NPC1 (0.51) NPC1RAB9ALMNACA2CTRB1
SCHEMBL9742824 0.81 NPC1 (0.51) NPC1RAB9ALMNACA2CTRB1
SCHEMBL7270681 0.78 CTRB1 (0.58) NPC1RAB9ALMNACTRB1
SCHEMBL1741997 0.77 NPC1 (0.60) NPC1RAB9A
SCHEMBL19954666 0.77 CTRB1 (0.54) NPC1RAB9ALMNACTRB1
SCHEMBL6445073 0.77 NPC1 (0.51) NPC1RAB9ALMNACA2CYP3A4
SCHEMBL6444710 0.77 NPC1 (0.51) NPC1RAB9ALMNACA2CYP3A4
SCHEMBL7332765 0.77 NPC1 (0.51) NPC1RAB9ALMNACA2CYP3A4
SCHEMBL6445202 0.77 NPC1 (0.51) NPC1RAB9ALMNACA2CYP3A4
SCHEMBL6931878 0.77 CTRB1 (0.59) NPC1RAB9ACTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed