SCHEMBL6448962

SCHEMBL6448962

CC(C)(C)NC(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)NC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
MAPT P10636 1/20 0.51
LMNA P02545 2/20 0.45
ALDH1A1 P00352 1/20 0.45
BCHE P06276 1/20 0.44
BACE1 P56817 2/20 0.43
CTRB1 P17538 1/20 0.42
MMP2 P08253 2/20 0.41
MMP3 P08254 1/20 0.41
CA2 P00918 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
KLK5 Q9Y337 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9742824 1.00 NPC1 (0.51) NPC1RAB9AMAPTLMNAALDH1A1
SCHEMBL7316559 0.86 BCHE (0.58) BCHEBACE1
SCHEMBL7302197 0.83 BCHE (0.55) BCHEBACE1
SCHEMBL6448790 0.81 NPC1 (0.60) NPC1RAB9ALMNACTRB1CA2
SCHEMBL8840299 0.80 BACE1 (0.40) NPC1RAB9AMAPTLMNAALDH1A1
SCHEMBL8432604 0.80 NAALAD2 (0.60) ALDH1A1
SCHEMBL7264947 0.80 NAALAD2 (0.60) ALDH1A1
SCHEMBL7547746 0.80 LAP3 (0.49) NPC1RAB9AMAPTLMNACTRB1
SCHEMBL6430008 0.80 LAP3 (0.49) NPC1RAB9AMAPTLMNACTRB1
SCHEMBL4957679 0.79 CA2 (0.43) NPC1RAB9AMAPTBCHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed