SCHEMBL6449677

SCHEMBL6449677

CCNC(=S)NC(CSC)C(=O)NCC#N.COc1ccc(NC(=S)NC(Cc2ccccc2)C(=O)NCC#N)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 3/20 0.52
CTSS P25774 8/20 0.49
CTSL P07711 8/20 0.49
CTSB P07858 5/20 0.49
CTSK P43235 5/20 0.48
RAB9A P51151 1/20 0.46
FPR1 P21462 2/20 0.45
MAOB P27338 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
TACR2 P21452 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6449673 0.92 FPR2 (0.47) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6818830 0.90 CTSL (0.54) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6019922 0.90 CTSL (0.60) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6020918 0.88 RAB9A (0.46) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6448627 0.86 CA1 (0.40) FPR2CTSSCTSLCTSBRAB9A
SCHEMBL6818828 0.84 FPR2 (0.48) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6020356 0.83 FPR2 (0.53) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6020012 0.82 CTSS (0.57) FPR2CTSSCTSLCTSBCTSK
SCHEMBL6019937 0.82 CTSS (0.70) CTSSCTSLCTSBCTSK
SCHEMBL6020162 0.81 CTSL (0.61) FPR2CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed