SCHEMBL6454902

SCHEMBL6454902

CCN(C(=O)c1ccc(C(=O)OC)s1)c1ccc(C)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 4/20 0.43
TSHR P16473 3/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HSD17B1 P14061 3/20 0.42
HSD17B2 P37059 3/20 0.42
LMNA P02545 1/20 0.41
PPARG P37231 1/20 0.41
NCOA2 Q15596 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
GAA P10253 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5557107 0.88 NPSR1 (0.43) ALDH1A1MAPTNPSR1TSHRHPGD
SCHEMBL5564443 0.88 NPSR1 (0.46) ALDH1A1MAPTNPSR1TSHRHPGD
SCHEMBL6455153 0.87 ALDH1A1 (0.50) ALDH1A1MAPTNPSR1TSHRHPGD
SCHEMBL5561977 0.83 ALDH1A1 (0.56) ALDH1A1MAPTNPSR1TSHRHPGD
SCHEMBL5559856 0.81 NPSR1 (0.40) ALDH1A1MAPTNPSR1TSHRHPGD
SCHEMBL5565995 0.80 KDM4E (0.48) ALDH1A1MAPTNPSR1TSHRHPGD
SCHEMBL5560541 0.80 SENP1 (0.43) ALDH1A1MAPTNPSR1L3MBTL1HSD17B1
SCHEMBL5560390 0.80 MAPKAPK2 (0.42) ALDH1A1MAPTL3MBTL1LMNATDP1
SCHEMBL5565065 0.78 NPSR1 (0.42) MAPTNPSR1TSHRHPGDMAPK1
SCHEMBL1588116 0.77 HPGD (0.51) ALDH1A1MAPTNPSR1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575933-A1 ENANTIOMERS OF THIOPHENE HYDROXAMIC ACID DERIVATIVES AND THEIR USE AS HDAC INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-09-21 EP disclosed
WO-2004054999-A1 ENANTIOMERS OF THIOPHENE HYDROXAMIC ACID DERIVATIVES AND THEIR USE AS HDAC INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-07-01 WO disclosed