SCHEMBL6454965

SCHEMBL6454965

NC(=O)c1cc(F)cc(OC2CCNCC2)c1F

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP2 Q9UGN5 3/20 0.49
PARP3 Q9Y6F1 2/20 0.49
MKNK1 Q9BUB5 2/20 0.48
MKNK2 Q9HBH9 2/20 0.48
MAP3K5 Q99683 1/20 0.45
HTR1A P08908 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
HRH1 P35367 1/20 0.38
PARP1 P09874 4/20 0.38
TOP2A P11388 3/20 0.38
HSP90AB1 P08238 2/20 0.38
UTS2R Q9UKP6 1/20 0.37
CHEK2 O96017 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6456150 0.84 MKNK1 (0.58) PARP2PARP3MKNK1MKNK2MAP3K5
SCHEMBL6454967 0.79 MKNK1 (0.49) PARP2PARP3MKNK1MKNK2MAP3K5
SCHEMBL4233748 0.74 MKNK1 (0.58) PARP2MKNK1MKNK2MAP3K5HTR1A
SCHEMBL6446339 0.73 MKNK1 (0.58) MKNK1MKNK2MAP3K5
SCHEMBL6451281 0.73 MKNK1 (0.58) MKNK1MKNK2MAP3K5HRH1TOP2A
SCHEMBL6447864 0.72 MKNK1 (0.46) PARP2PARP3MKNK1MKNK2MAP3K5
SCHEMBL6447886 0.72 OPRM1 (0.54) MKNK1MKNK2MAP3K5HTR1ASLC6A2
SCHEMBL16828784 0.72 MKNK1 (0.51) MKNK1MKNK2MAP3K5TOP2AHSP90AB1
SCHEMBL6450115 0.72 MAP3K5 (0.47) PARP2PARP3MKNK1MKNK2MAP3K5
SCHEMBL5372678 0.72 MKNK1 (0.51) MKNK1MKNK2MAP3K5HRH1TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6964974-B2 2,3-oxidosqualene-lanosterol cyclase inhibitors HOFFMANN-LA ROCHE INC. (US) 2005-11-15 US disclosed