SCHEMBL6454967

SCHEMBL6454967

NC(=O)c1cc(F)c(OC2CCNCC2)cc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 2/20 0.49
MKNK2 Q9HBH9 2/20 0.49
MAP3K5 Q99683 1/20 0.46
ROCK2 O75116 1/20 0.45
HTR1A P08908 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A3 Q01959 2/20 0.43
PARP2 Q9UGN5 2/20 0.41
PARP3 Q9Y6F1 2/20 0.41
SCN9A Q15858 1/20 0.39
PARP1 P09874 1/20 0.39
TOP2A P11388 3/20 0.38
HSP90AB1 P08238 2/20 0.38
BCL9 O00512 1/20 0.37
CTNNB1 P35222 1/20 0.37
CHEK2 O96017 1/20 0.37
NTRK1 P04629 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6456150 0.80 MKNK1 (0.58) MKNK1MKNK2MAP3K5HTR1ASLC6A2
SCHEMBL6447886 0.79 OPRM1 (0.54) MKNK1MKNK2MAP3K5HTR1ASLC6A2
SCHEMBL6454965 0.79 PARP2 (0.49) MKNK1MKNK2MAP3K5HTR1ASLC6A2
Hydrochloric Acid SCHEMBL31753763 0.77 SCN9A (0.54) ROCK2SCN9APARP1CHEK2
SCHEMBL6154865 0.75 ROCK2 (0.72) ROCK2PARP2PARP3PARP1
SCHEMBL4233748 0.75 MKNK1 (0.58) MKNK1MKNK2MAP3K5HTR1ASLC6A2
SCHEMBL6446339 0.74 MKNK1 (0.58) MKNK1MKNK2MAP3K5
SCHEMBL6451281 0.74 MKNK1 (0.58) MKNK1MKNK2MAP3K5TOP2AHSP90AB1
SCHEMBL17062481 0.74 SCN9A (0.49) HTR1ASLC6A2SLC6A3SCN9A
SCHEMBL6447882 0.73 HTR1A (0.56) MKNK1MKNK2MAP3K5HTR1ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6964974-B2 2,3-oxidosqualene-lanosterol cyclase inhibitors HOFFMANN-LA ROCHE INC. (US) 2005-11-15 US disclosed