SCHEMBL6455092

SCHEMBL6455092

C#CCOC(OCC#C)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 1/20 0.35
HTR2A P28223 2/20 0.34
TAAR1 Q96RJ0 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2D6 P10635 3/20 0.34
TSHR P16473 3/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAOB P27338 3/20 0.33
SCN1A P35498 2/20 0.33
SCN2A Q99250 2/20 0.33
SCN3A Q9NY46 2/20 0.33
MAOA P21397 1/20 0.33
LMNA P02545 1/20 0.33
CHRM2 P08172 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28821628 0.88 KMT2A (0.36) NPC1MEN1KMT2AMAPTHTR2A
SCHEMBL26661470 0.84 NPC1 (0.35) NPC1MEN1KMT2ACYP1A2CYP2D6
SCHEMBL17288627 0.83 MEN1 (0.51) MEN1KMT2AHTR2ASMN1; SMN2CYP1A2
SCHEMBL3175966 0.81 CYP3A4 (0.44) NPC1MEN1KMT2ACYP1A2CYP2D6
SCHEMBL11555379 0.81 PPARG (0.38) TSHRMAOA
SCHEMBL10346414 0.79 CYP1A2 (0.38) NPC1MEN1KMT2AHTR2ATAAR1
SCHEMBL76084 0.79 LMNA (0.38) MEN1KMT2ASMN1; SMN2TSHRCYP2C9
SCHEMBL8749377 0.79 NPC1 (0.40) NPC1MEN1KMT2ACYP1A2CYP2D6
SCHEMBL11314272 0.79 PYCR1 (0.35) NPC1MEN1KMT2ASMN1; SMN2CYP1A2
SCHEMBL27811527 0.79 TRPA1 (0.38) NPC1MEN1KMT2AMAPTHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546371-A1 SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (EPFL) (CH) 2005-06-29 EP disclosed
WO-2004031405-A1 SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (EPFL) (CH) 2004-04-15 WO disclosed