SCHEMBL6461487

SCHEMBL6461487

COc1ccc(C[C@@](N)(CC(=O)O)c2ccccc2)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
HTT P42858 1/20 0.48
LDHA P00338 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 3/20 0.44
LMNA P02545 1/20 0.44
KIF11 P52732 1/20 0.44
GAA P10253 2/20 0.43
KMT2A Q03164 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
MEN1 O00255 1/20 0.43
PRKCZ Q05513 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP19A1 P11511 1/20 0.42
REN P00797 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706894 0.75 SMN1; SMN2 (0.56) SMN1; SMN2HTTLDHACYP1A2CYP3A4
SCHEMBL6339567 0.75 ALDH1A1 (0.60) HTTLDHACYP1A2CYP3A4CYP2C19
SCHEMBL29658682 0.75 ALDH1A1 (0.60) HTTLDHACYP1A2CYP3A4CYP2C19
SCHEMBL29658681 0.75 ALDH1A1 (0.60) HTTLDHACYP1A2CYP3A4CYP2C19
SCHEMBL6339568 0.75 ALDH1A1 (0.60) HTTLDHACYP1A2CYP3A4CYP2C19
SCHEMBL24534351 0.75 ALDH1A1 (0.60) HTTLDHACYP1A2CYP3A4CYP2C19
SCHEMBL8550004 0.73 L3MBTL1 (0.46) SMN1; SMN2HTTCYP1A2ALDH1A1LMNA
Hydrochloric Acid SCHEMBL29152364 0.73 ALDH1A1 (0.59) HTTLDHACYP1A2CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL30149960 0.73 ALDH1A1 (0.59) HTTLDHACYP1A2CYP3A4CYP2C19
SCHEMBL27986995 0.73 ALDH1A1 (0.59) HTTLDHACYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493819-B1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER UBE INDUSTRIES (JP) 2014-11-12 EP disclosed
EP-1493819-A1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER Ube Industries, Ltd. (JP) 2005-01-05 EP disclosed