SCHEMBL6461819

SCHEMBL6461819

CC(CCNC(=O)O)CC(=O)NCCC(C(=O)c1nc(C(=O)NCC23CC4CC(CC(C4)C2)C3)co1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.39
CTSL P07711 1/20 0.37
TP53 P04637 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
CNR1 P21554 1/20 0.33
ABCB11 O95342 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7047185 0.90 CTSL (0.37) P2RX7CTSLALDH1A1EPHX2
SCHEMBL7567547 0.84 ALDH1A1 (0.35) MEN1ALDH1A1KMT2AEPHX2
SCHEMBL6467927 0.81 GAA (0.44) MEN1ALDH1A1KMT2A
SCHEMBL6467203 0.78 SMN1; SMN2 (0.35) MEN1ALDH1A1KMT2AEPHX2
SCHEMBL7049037 0.72 KCNA5 (0.39) ALDH1A1
SCHEMBL6475534 0.72 SMN1; SMN2 (0.39) MEN1ALDH1A1KMT2A
SCHEMBL7049297 0.72 HPGD (0.40) MEN1ALDH1A1KMT2A
SCHEMBL7047980 0.72 TBXA2R (0.37) MEN1ALDH1A1KMT2ACNR1
SCHEMBL7046299 0.71 L3MBTL1 (0.44) ALDH1A1KMT2AEPHX2
SCHEMBL7044845 0.71 KCNA5 (0.39) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed