SCHEMBL6462828

SCHEMBL6462828

CCC[C@H](NC(=O)N(CCS(=O)(=O)Cc1ccccc1OC)C(=O)O)C(=O)c1nc2ccccc2o1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CTSK P43235 1/20 0.38
XDH P47989 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7043205 0.94 CTSS (0.39) CTSSCYP3A4CYP2C9CTSKXDH
SCHEMBL6468436 0.88 CTSS (0.44) CTSSCYP3A4CYP2C9XDH
SCHEMBL6466173 0.88 CTSS (0.39) CTSSCYP3A4CYP2C9
SCHEMBL6462867 0.84 CTSS (0.41) CTSSCYP3A4CYP2C9XDH
SCHEMBL6464424 0.82 CTSS (0.43) CTSSCYP3A4CYP2C9XDH
SCHEMBL6464410 0.82 FAAH (0.42) CTSSCYP3A4CYP2C9CTSK
SCHEMBL6467432 0.81 P2RY14 (0.37) CTSSCYP3A4CYP2C9CTSK
SCHEMBL6462825 0.80 XDH (0.38) CYP3A4XDH
SCHEMBL6463818 0.80 CTSS (0.40) CTSSCYP3A4CYP2C9CTSK
SCHEMBL7046394 0.79 CTSS (0.40) CTSSCYP3A4CYP2C9XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed