SCHEMBL6464410

SCHEMBL6464410

O=C(c1nc2ccccc2o1)[C@H](CCc1ccccc1)NC(=O)N(CCS(=O)(=O)Cc1ccccc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.42
CES1 P23141 1/20 0.42
DAGLA Q9Y4D2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CTSS P25774 16/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41
CTSK P43235 2/20 0.41
PRSS8 Q16651 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468436 0.92 CTSS (0.44) ALDH1A1CTSSCYP3A4CYP2C9
SCHEMBL6464424 0.91 CTSS (0.43) ALDH1A1CTSSCYP3A4CYP2C9
SCHEMBL6475526 0.86 FAAH (0.46) FAAHCES1DAGLACTSSCYP3A4
SCHEMBL6466984 0.86 PRSS8 (0.41) CTSSCYP3A4CYP2C9CTSLCTSB
SCHEMBL6062110 0.86 CTSS (0.37) FAAHCES1DAGLACTSSCYP3A4
SCHEMBL6462867 0.85 CTSS (0.41) ALDH1A1CTSSCYP3A4CYP2C9
SCHEMBL7046394 0.84 CTSS (0.40) ALDH1A1CTSSCYP3A4CYP2C9PRSS8
SCHEMBL6467558 0.83 FAAH (0.46) FAAHCES1DAGLACTSSCYP3A4
SCHEMBL6462828 0.82 CTSS (0.41) CTSSCYP3A4CYP2C9CTSK
SCHEMBL6465390 0.82 ALDH1A1 (0.41) FAAHCES1DAGLAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed