SCHEMBL646485

SCHEMBL646485

CN(C)C(c1ccccc1)C1CCC(NC(=O)CCCCCN(C)S(=O)(=O)c2c(Cl)cc(Cl)cc2Cl)CC1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
FASN P49327 1/20 0.39
ICMT O60725 1/20 0.36
ALB P02768 1/20 0.36
HDAC3 O15379 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC6 Q9UBN7 3/20 0.36
POLB P06746 1/20 0.35
BDKRB1 P46663 1/20 0.35
EPHX1 P07099 1/20 0.35
ENPP2 Q13822 1/20 0.35
CNR2 P34972 1/20 0.34
CNR1 P21554 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTR4 Q13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL643276 0.99 BCHE (0.38) BCHEACHEFASNICMTALB
SCHEMBL645438 0.88 HDAC3 (0.37) HDAC3HDAC1HDAC2HDAC6CNR2
SCHEMBL2489242 0.88 ICMT (0.35) ICMTALBCNR2CNR1
SCHEMBL644640 0.87 HDAC3 (0.36) HDAC3HDAC1HDAC2HDAC6CNR2
SCHEMBL492647 0.86 RAB9A (0.34) POLBRAB9AALDH1A1
SCHEMBL492815 0.86 BDKRB1 (0.36) POLBBDKRB1ALDH1A1
SCHEMBL644329 0.85 CACNA2D1 (0.37) BCHEACHEICMTALBHDAC3
SCHEMBL493265 0.81 BDKRB1 (0.35) POLBBDKRB1ALDH1A1
SCHEMBL2489881 0.80 LMNA (0.35) CNR2CNR1RAB9AALDH1A1
SCHEMBL492775 0.79 ALDH1A1 (0.37) POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119633-B2 N-{2-[2-(4-benzyl-4-hydroxy-piperidin-1-yl)-2-oxo-ethoxy]-ethyl}-N-ethyl-4-methoxy-2,3,6-trimethyl-phenylsulfonamide; condensing the N-carboxyalkyl phenylsulfonamide with the substituted piperidine; bradykinin receptor antagonists; analgesics; antidiabetics; angiogenesis inhibitors; rheumatic diseases GRUENENTHAL GMBH (DE) 2012-02-21 US claimed