SCHEMBL6466262

SCHEMBL6466262

CC1CCN(CC(N2CCC(C)CC2)n2c(=O)oc3ccccc32)CC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PLD1 Q13393 1/20 0.41
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7062216 0.86 SIGMAR1 (0.48) MEN1KMT2A
SCHEMBL6460781 0.85 CHRM1 (0.39) PLD1
SCHEMBL2150109 0.74 MEN1 (0.64) MEN1KMT2A
SCHEMBL2149712 0.72 CHRM1 (0.63)
SCHEMBL2149643 0.72 HTR1A (0.66)
SCHEMBL6462861 0.69 POLB (0.50) MEN1KMT2AMAPK1
SCHEMBL29591678 0.67 MAPK1 (0.52) MEN1KMT2AMAPK1
SCHEMBL2600306 0.67 MAPK1 (0.52) MEN1KMT2AMAPK1
SCHEMBL16997531 0.66 TNKS (0.57) MEN1KMT2APLD1MAPK1
SCHEMBL6454535 0.65 SIGMAR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432420-A4 BENZIMIDAZOLIDINONE DERIVATIVES AS MUSCARINIC AGENTS ACADIA PHARM INC (US) 2005-11-09 EP disclosed
EP-1432420-A2 BENZIMIDAZOLIDINONE DERIVATIVES AS MUSCARINIC AGENTS Acadia Pharmaceuticals Inc. (US) 2004-06-30 EP disclosed
WO-2003028650-A2 BENZIMIDAZOLIDINONE DERIVATIVES AS MUSCARINIC AGENTS ACADIA PHARMACEUTICALS, INC. (US) 2003-04-10 WO disclosed