SCHEMBL6467749

SCHEMBL6467749

COc1ccc2c(c1)C[C@@H](C)[C@@H]1[C@@H]2CC[C@]2(C)C(CO[Si](C)(C)C(C)(C)C)=CC[C@H]12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.39
HSD17B1 P14061 2/20 0.38
LMNA P02545 4/20 0.38
MAPT P10636 1/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ESR1 P03372 8/20 0.38
ESR2 Q92731 2/20 0.38
STS P08842 2/20 0.37
HSD17B10 Q99714 1/20 0.36
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
CNR1 P21554 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6462339 0.84 ESR1 (0.51) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL4370456 0.80 LMNA (0.42) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6462626 0.78 STS (0.42) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6468153 0.78 LMNA (0.41) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6464758 0.76 HRH3 (0.39) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL7704384 0.76 HRH3 (0.39) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6569627 0.73 HRH3 (0.39) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6464576 0.73 HSD17B1 (0.38) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6569630 0.73 HRH3 (0.39) HRH3HSD17B1LMNAMAPTRECQL
SCHEMBL6527877 0.73 LMNA (0.41) HRH3HSD17B1LMNAMAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6881728-B1 14-β, 17-α-hydroxymethylandrostane derivatives as androgens AKZO NOBEL N.V. (NL) 2005-04-19 US disclosed
EP-1163259-A1 14.BETA.,17-ALPHA-HYDROXYMETHYLANDROSTANE DERIVATIVES AS ANDROGENS Akzo Nobel N.V. (NL) 2001-12-19 EP disclosed
WO-2000053619-A1 14.BETA., 17-ALPHA-HYDROXYMETHYLANDROSTANE DERIVATIVES AS ANDROGENS AKZO NOBEL N.V. (NL) 2000-09-14 WO disclosed