SCHEMBL6469128

SCHEMBL6469128

CSc1ccc(-c2[nH]nc(N(C=O)CCO)c2C2CCCCC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
JAK2 O60674 2/20 0.33
JAK1 P23458 2/20 0.33
TYK2 P29597 2/20 0.33
JAK3 P52333 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6438697 0.86 PTGS2 (0.40) JAK2JAK1TYK2JAK3
SCHEMBL6437926 0.81 PTGS2 (0.39) JAK2JAK1TYK2JAK3
SCHEMBL6440473 0.74 GAA (0.43) GAA
SCHEMBL6442323 0.72 GAA (0.40) GAA
SCHEMBL6444360 0.71 ALDH1A1 (0.36) GAA
SCHEMBL5150592 0.71 ALDH1A1 (0.36) GAA
SCHEMBL3866503 0.67 PTGS2 (0.39)
SCHEMBL4957820 0.65 CDK1 (0.36) GAA
SCHEMBL3864227 0.62 PTGS2 (0.38)
SCHEMBL6438872 0.62 PTGS2 (0.47) JAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed