Anthranilamide

Anthranilamide

SCHEMBL6469157

CCCCCOc1ccc2[nH]c(C(=O)O)cc2c1.NC(=O)c1ccccc1N

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G4A P47712 1/20 0.54
ALDH1A1 P00352 4/20 0.54
KDM4E B2RXH2 3/20 0.54
HSD17B10 Q99714 3/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
HPGD P15428 1/20 0.54
SRD5A2 P31213 1/20 0.54
PDGFRB P09619 6/20 0.49
PDGFRA P16234 6/20 0.49
CFD P00746 1/20 0.49
KMT2A Q03164 2/20 0.49
PTPN11 Q06124 1/20 0.47
MAPT P10636 2/20 0.45
MEN1 O00255 1/20 0.45
NR1I2 O75469 1/20 0.45
LMNA P02545 1/20 0.45
CHRM2 P08172 1/20 0.45
CYP3A4 P08684 1/20 0.45
ADRA2A P08913 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6469163 0.92 KDM4E (0.60) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL4360657 0.86 PLA2G4A (0.68) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL4369016 0.84 PLA2G4A (0.67) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
Anthranilamide SCHEMBL6335928 0.83 HSD17B10 (0.55) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL1144832 0.79 KDM4E (0.65) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL6469159 0.79 HDAC1 (0.63) ALDH1A1KDM4EPDGFRBPDGFRAMAPT
SCHEMBL9816433 0.77 KDM4E (0.73) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL13174431 0.74 KDM4E (0.62) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL24076666 0.74 PLA2G4A (0.55) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2
SCHEMBL2767179 0.74 KDM4E (0.65) PLA2G4AALDH1A1KDM4EHSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2005508311-A 2005-03-31 JP claimed
EP-1416928-A2 N-MONOACYLATED DERIVATIVES OF O-PHENYLENEDIAMINES, THEIR SIX MEMBERED HETEROCYCLIC ANALOGUES AND THEIR USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2004-05-12 EP claimed
WO-2003013484-A2 N-MONOACYLATED DERIVATIVES OF O-PHENYLENEDIAMINES, THEIR SIX MEMBERED HETEROCYCLIC ANALOGUES AND THEIR USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2003-02-20 WO claimed