SCHEMBL6469289

SCHEMBL6469289

CC1=C(C)C(C)C([Ti](C)(C)NC(=O)C2CCCCCCCCCCC2)=C1C.[SiH4]

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
P2RX7 Q99572 2/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 2/20 0.33
MAPK1 P28482 2/20 0.33
CYP3A4 P08684 1/20 0.33
PTPN1 P18031 1/20 0.33
HPGD P15428 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7622820 1.00 HDAC8 (0.36) HDAC8HDAC6KMT2AMEN1LMNA
SCHEMBL727844 0.99 HDAC8 (0.37) HDAC8HDAC6KMT2AMEN1LMNA
SCHEMBL5968790 0.88
SCHEMBL5968791 0.88
SCHEMBL5968778 0.85 HPGD (0.37) HDAC8HDAC6LMNARAB9ASMN1; SMN2
SCHEMBL5969036 0.85 HPGD (0.37) HDAC8HDAC6LMNARAB9ASMN1; SMN2
SCHEMBL7246533 0.76 P2RX7 (0.38) KMT2ALMNANPSR1RAB9ASMN1; SMN2
SCHEMBL7679958 0.74
SCHEMBL7924767 0.71 ALDH1A1 (0.33) KMT2ARAB9ASMN1; SMN2NPC1TSHR
SCHEMBL8073123 0.68 KMT2A (0.40) HDAC8HDAC6KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1509552-A1 SOLID, PARTICULATED, SPRAY DRIED, HETEROGENOUS CATALYST COMPOSITION Univation Technologies LLC (US) 2005-03-02 EP disclosed
EP-1412365-A1 SALT OF LEWIS ACID/ACID ADDUCTS AND CATALYST ACTIVATORS THEREFROM DOW GLOBAL TECHNOLOGIES INC. (US) 2004-04-28 EP disclosed
US-6727329-B2 USEFUL IN SOLUTION, GAS PHASE, SLURRY AND CATIONIC POLYMERIZATION OF OLEFINS DOW GLOBAL TECHNOLOGY INC. 2004-04-27 US disclosed
WO-2003102037-A1 SOLID, PARTICULATED, SPRAY DRIED, HETEROGENOUS CATALYST COMPOSITION UNIVATION TECHNOLOGIES, LLC (US) 2003-12-11 WO disclosed
WO-2003010171-A1 SALT OF LEWIS ACID/ACID ADDUCTS AND CATALYST ACTIVATORS THEREFROM DOW GLOBAL TECHNOLOGIES, INC. (US) 2003-02-06 WO disclosed
EP-1259556-A2 IMPROVED SILANE FUNCTIONALIZED OLEFIN INTERPOLYMERS AND DERIVATIVES THEREOF THE DOW CHEMICAL COMPANY (US) 2002-11-27 EP disclosed
US-20020132729-A1 Catalyst activators comprising expanded anions LAPOINTE ROBERT E (US) 2002-09-19 US disclosed
EP-1228109-A1 SUPPORTED CATALYST COMPRISING EXPANDED ANIONS THE DOW CHEMICAL COMPANY (US) 2002-08-07 EP disclosed
WO-2002008303-A1 EXPANDED ANIONIC COMPOUNDS COMPRISING HYDROXYL OR QUIESCENT REACTIVE FUNCTIONALITY AND CATALYST ACTIVATORS THEREFROM THE DOW CHEMICAL COMPANY (US) 2002-01-31 WO disclosed
WO-2001023442-A1 SUPPORTED CATALYST COMPRISING EXPANDED ANIONS THE DOW CHEMICAL COMPANY (US) 2001-04-05 WO disclosed
WO-2001009207-A2 IMPROVED SILANE FUNCTIONALIZED OLEFIN INTERPOLYMERS AND DERIVATIVES THEREOF THE DOW CHEMICAL COMPANY (US) 2001-02-08 WO disclosed
EP-1056752-A1 CATALYST ACTIVATORS COMPRISING EXPANDED ANIONS THE DOW CHEMICAL COMPANY (US) 2000-12-06 EP disclosed
EP-1054910-A1 IMPROVED OLEFIN POLYMERIZATION PROCESS THE DOW CHEMICAL COMPANY (US) 2000-11-29 EP disclosed
WO-1999042467-A1 CATALYST ACTIVATORS COMPRISING EXPANDED ANIONS THE DOW CHEMICAL COMPANY (US) 1999-08-26 WO disclosed
WO-1999041289-A1 IMPROVED OLEFIN POLYMERIZATION PROCESS THE DOW CHEMICAL COMPANY (US) 1999-08-19 WO disclosed