SCHEMBL6471830

SCHEMBL6471830

C=CCCOC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)N(C#N)S(C)(=O)=O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NMBR P28336 10/20 0.49
TACR1 P25103 3/20 0.47
CTSL P07711 2/20 0.47
CTSS P25774 1/20 0.47
CTSK P43235 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
MMP14 P50281 1/20 0.45
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
CCKBR P32239 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6020424 0.88 NMBR (0.52) NMBRTACR1CTSLCTSSCTSK
SCHEMBL6019136 0.87 NMBR (0.51) NMBRTACR1CTSLCTSSCTSK
SCHEMBL6020423 0.82 CTSL (0.69) NMBRTACR1CTSLCTSSCTSK
SCHEMBL6019145 0.81 NMBR (0.58) NMBRTACR1CTSLCTSSCTSK
SCHEMBL6471832 0.81 NMBR (0.56) NMBRTACR1CTSLCTSSCTSK
SCHEMBL6019142 0.79 NMBR (0.65) NMBRTACR1CTSLCTSSCTSK
SCHEMBL732867 0.76 ALOX15 (0.59) NMBRTACR1ALOX15
SCHEMBL6020520 0.76 CCKBR (0.55) NMBRTACR1CTSLCTSSCTSK
SCHEMBL6020206 0.76 NMBR (0.53) NMBRCTSLCTSSCTSKKDM4E
SCHEMBL6020369 0.75 NMBR (0.65) NMBRTACR1CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed