SCHEMBL6471832

SCHEMBL6471832

C=CCCOC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)NS(=O)(=O)CC#N

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NMBR P28336 12/20 0.56
CTSL P07711 2/20 0.51
CTSS P25774 1/20 0.51
CTSK P43235 1/20 0.51
MAPT P10636 3/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TACR1 P25103 1/20 0.49
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46
TACR3 P29371 1/20 0.45
CA2 P00918 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6020423 0.86 CTSL (0.69) NMBRCTSLCTSSCTSKMAPT
SCHEMBL6019142 0.84 NMBR (0.65) NMBRCTSLCTSSCTSKMAPT
SCHEMBL6019145 0.83 NMBR (0.58) NMBRCTSLCTSSCTSKMAPT
SCHEMBL6471830 0.81 NMBR (0.49) NMBRCTSLCTSSCTSKMAPT
SCHEMBL6020424 0.80 NMBR (0.52) NMBRCTSLCTSSCTSKMAPT
SCHEMBL6019136 0.79 NMBR (0.51) NMBRCTSLCTSSCTSKMAPT
SCHEMBL732867 0.76 ALOX15 (0.59) NMBRTACR1
SCHEMBL10888014 0.74 ALOX15 (0.64) NMBR
SCHEMBL28836525 0.74 ALOX15 (0.64) NMBR
SCHEMBL29908071 0.74 ALOX15 (0.64) NMBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed