SCHEMBL6473206

SCHEMBL6473206

CS(=O)(=O)C1(S(C)(=O)=O)C2CCC1(CS(=O)(=O)NC(Cc1csc3ccccc13)C(=O)NCCC#N)C(=O)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
MMP2 P08253 3/20 0.38
MMP9 P14780 3/20 0.38
MMP8 P22894 3/20 0.38
MMP1 P03956 2/20 0.38
ITGB3 P05106 2/20 0.36
ITGAV P06756 2/20 0.36
CYP2C19 P33261 2/20 0.34
CYP1A2 P05177 1/20 0.34
F10 P00742 1/20 0.34
DPP4 P27487 2/20 0.33
DPP8 Q6V1X1 2/20 0.33
DPP9 Q86TI2 2/20 0.33
CASP1 P29466 1/20 0.33
MMP3 P08254 1/20 0.33
MMP14 P50281 1/20 0.33
MMP25 Q9NPA2 1/20 0.33
MTNR1A P48039 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6020361 0.91 MMP1 (0.45) CTSLCTSSCTSKMMP2MMP9
SCHEMBL6020368 0.85 CTSL (0.51) CTSLCTSSCTSKMMP2MMP9
SCHEMBL6473203 0.84 CTSL (0.38) CTSLCTSSCTSKMMP2MMP9
SCHEMBL6020996 0.77 MMP1 (0.45) CTSLCTSSCTSKMMP2MMP9
SCHEMBL6019805 0.77 MMP1 (0.57) MMP2MMP9MMP8MMP1ITGB3
SCHEMBL6020634 0.76 MMP1 (0.44) CTSLCTSSCTSKMMP2MMP9
SCHEMBL6021301 0.74 ITGB3 (0.55) CTSSCTSKMMP2MMP9MMP8
SCHEMBL6020633 0.73 CTSL (0.53) CTSLCTSSCTSKMMP2MMP9
SCHEMBL6019703 0.73 ITGB3 (0.54) MMP2MMP9MMP8MMP1ITGB3
SCHEMBL6020883 0.72 ALDH1A1 (0.47) MMP2MMP9MMP8MMP1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed