SCHEMBL6473349

SCHEMBL6473349

Cc1ccc(CC(C)(C)[C@H]2Cc3ccccc3O2)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.37
MAOB P27338 6/20 0.37
TSHR P16473 1/20 0.36
HIF1A Q16665 3/20 0.36
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
SSTR4 P31391 1/20 0.34
AOC2 O75106 5/20 0.33
MAOA P21397 5/20 0.33
DAO P14920 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
HRH1 P35367 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6477728 1.00 CYP19A1 (0.37) CYP19A1MAOBTSHRHIF1AALDH1A1
SCHEMBL11952613 0.74 SSTR4 (0.41) MAOBTSHRHIF1ASSTR4AOC2
SCHEMBL10877666 0.72 HIF1A (0.52) HIF1AALDH1A1SSTR4
SCHEMBL8035974 0.72 AOC2 (0.40) MAOBTSHRHIF1ASSTR4AOC2
SCHEMBL10366394 0.69 HIF1A (0.38) CYP19A1MAOBTSHRHIF1ASSTR4
SCHEMBL8036060 0.69 SSTR4 (0.43) MAOBHIF1ASSTR4AOC2MAOA
SCHEMBL5777888 0.69 PPARG (0.41) TSHRHIF1AALDH1A1SSTR4MAPT
SCHEMBL23625404 0.69 ALDH1A1 (0.33) HIF1AALDH1A1
SCHEMBL23645657 0.69 TDP1 (0.42) HIF1AALDH1A1RAB9AMAPT
SCHEMBL7279348 0.68 SSTR4 (0.45) MAOBTSHRHIF1AALDH1A1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005012209-A2 CATALYZED ENANTIOSELECTIVE TRANSFORMATION OF ALKENES UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2005-02-10 WO claimed
WO-2005012209-A2 CATALYZED ENANTIOSELECTIVE TRANSFORMATION OF ALKENES UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2005-02-10 WO disclosed