Bromide

Bromide

SCHEMBL6474963

Br.Nc1ccc(Cl)cc1CBr

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.50
TSHR P16473 3/20 0.50
ALOX15 P16050 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
ALDH1A1 P00352 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
TP53 P04637 1/20 0.43
HPGD P15428 2/20 0.40
ALOX12 P18054 2/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
IDO1 P14902 5/20 0.39
KMT2A Q03164 2/20 0.39
HIF1A Q16665 2/20 0.39
MEN1 O00255 1/20 0.39
SLC22A1 O15245 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
HSP90AA1 P07900 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6484010 0.83 CYP3A4 (0.50) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL14085079 0.80 CYP3A4 (0.52) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL775188 0.77 CYP3A4 (0.54) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL384040 0.77 IDO1 (0.44) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL30089455 0.77 IDO1 (0.44) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL6055610 0.76 CYP3A4 (0.52) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL775187 0.76 CYP3A4 (0.52) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL3786384 0.76 CYP3A4 (0.52) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL703030 0.76 CYP3A4 (0.52) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1
SCHEMBL23435078 0.75 CYP3A4 (0.46) CYP3A4TSHRALOX15SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6906078-B2 Method of using (H+/K+) ATPase inhibitors as antiviral agents PHARMACIA CORPORATION (US) 2005-06-14 US disclosed
US-20010047038-A1 Method of using (H+/K+) ATPase inhibitors as antiviral agents MOORMAN ALAN E (US) 2001-11-29 US disclosed
US-5945425-A ADENOSINE TRIPHOSPHASE INHIBITOR; DNA VIRICIDE G.D. SEARLE & CO. (US) 1999-08-31 US disclosed
US-5869513-A ANTIULCER AGENTS G. D. SEARLE & CO. (US) 1999-02-09 US disclosed
WO-1995029897-A1 METHOD OF USING (H+/K+) ATPase INHIBITORS AS ANTIVIRAL AGENTS G.D. SEARLE & CO. (US) 1995-11-09 WO disclosed
EP-0204215-A1 2-[(1H-benzimidazol-2-ylsulfinyl)methyl]-benzenamines G.D. Searle & Co. (US) 1986-12-10 EP disclosed
US-4214889-A Benzoxazine herbicides SANDOZ, INC. (US) 1980-07-29 US disclosed
US-4164407-A Benzoxazine herbicides SANDOZ, INC. (US) 1979-08-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010047038-A1 Method of using (H+/K+) ATPase inhibitors as antiviral agents ATP4A, ATP1A1, ATP1A4 CYP3A4 1001/4885TSHR 3552/4885ALOX15 3259/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.