SCHEMBL6477306

SCHEMBL6477306

N#Cc1ccc(CNC(=O)[C@H]2CCCN2C(=O)CNC2CCCCC2)cn1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
DPP4 P27487 11/20 0.47
DPP8 Q6V1X1 2/20 0.45
DPP9 Q86TI2 2/20 0.45
NAMPT P43490 1/20 0.44
F2 P00734 2/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
CYP2C19 P33261 1/20 0.41
FAP Q12884 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6483096 0.83 F2 (0.53) ALDH1A1NAMPTF2CYP3A4CYP2C9
SCHEMBL6476398 0.81 F2 (0.51) ALDH1A1F2FAP
SCHEMBL6487152 0.81 NAMPT (0.48) ALDH1A1NAMPTCYP3A4CYP2C9PKM
Acetic Acid SCHEMBL6484260 0.80 F2 (0.50) ALDH1A1NAMPTF2CYP3A4CYP2C9
SCHEMBL6477216 0.80 ALDH1A1 (0.50) ALDH1A1F2CYP3A4CYP2C9PKM
SCHEMBL8301494 0.79 F2 (0.48) ALDH1A1DPP4NAMPTF2CYP3A4
SCHEMBL6476709 0.79 ALDH1A1 (0.47) ALDH1A1NAMPTF2CYP3A4CYP2C9
SCHEMBL6487234 0.78 F2 (0.52) ALDH1A1F2
SCHEMBL23752337 0.77 F2 (0.69) ALDH1A1F2
SCHEMBL21067875 0.77 F2 (0.69) ALDH1A1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900319-B2 Thrombin inhibitors ABBOTT GMBH & CO. KG (DE) 2005-05-31 US disclosed
US-20020169318-A1 Novel thrombin inhibitors ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2002-11-14 US disclosed
US-6444817-B1 ANTICOAGULANTS ABBOTT LABORATORIES 2002-09-03 US disclosed
US-6030972-A 2- OR 5-AMINOMETHYL,2- OR 5-CYANOPYRIMIDINES AS INTERMEDIATES OF ANTICOAGULANTS IN EXTRACORPOREAL CIRCULATION (HEART-LUNG MACHINE, HEMODIALYSIS) BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169318-A1 Novel thrombin inhibitors TFPI, SERPINC1, F11 ALDH1A1 925/4885DPP4 551/4885DPP8 346/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.