SCHEMBL6478605

SCHEMBL6478605

O=[C]c1ccc(C2=CCOc3ccccc32)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 5/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
KDM4E B2RXH2 2/20 0.30
GLA P06280 2/20 0.30
GAA P10253 1/20 0.30
PIM1 P11309 1/20 0.30
ATM Q13315 1/20 0.30
CYP19A1 P11511 1/20 0.30
KMT2A Q03164 1/20 0.30
KCNH2 Q12809 3/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1354897 0.81 OPRD1 (0.41) OPRD1PKMTSHRKDM4EGAA
SCHEMBL6478611 0.78 ELANE (0.39) PKMTSHRKMT2A
SCHEMBL6491384 0.77 OPRD1 (0.51) OPRD1TSHRKCNH2OPRK1
SCHEMBL6492765 0.76 OPRD1 (0.39) OPRD1PKMTSHRKCNH2OPRK1
SCHEMBL2004582 0.73 TSHR (0.42) PKMTSHRKDM4EGLAGAA
SCHEMBL6480972 0.73 OPRD1 (0.55) OPRD1TSHRKDM4EGLAGAA
SCHEMBL8657572 0.68 PKM (0.42) PKMTSHRCYP19A1KMT2A
SCHEMBL7039789 0.66 PKM (0.42) PKMTSHRKDM4EGAACYP19A1
SCHEMBL276292 0.66 PKM (0.47) PKMTSHRCYP19A1KMT2A
SCHEMBL7430943 0.66 PKM (0.39) PKMTSHRCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6962938-B2 Spiro-cyclic β-amino acid derivatives as inhibitors of matrix metalloproteases and TNF-α converting enzyme (TACE) BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2005-11-08 US disclosed
US-6720329-B2 ANTIINFLAMMATORY AGENTS BRISTOL-MYERS SQUIBB PHARMA 2004-04-13 US disclosed