SCHEMBL6482379

SCHEMBL6482379

O=S(=O)(Nc1cccc(CCOCc2csc(-c3ccc(Cl)cc3)n2)c1)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 1/20 0.43
KDM1A O60341 1/20 0.43
GPR119 Q8TDV5 1/20 0.42
MAPT P10636 8/20 0.42
RHOC P08134 1/20 0.41
RHOA P61586 1/20 0.41
TP53 P04637 4/20 0.41
PPARA Q07869 2/20 0.41
PPARG P37231 1/20 0.41
LMNA P02545 3/20 0.40
GFER P55789 1/20 0.40
CYSLTR2 Q9NS75 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6475724 0.92 TP53 (0.42) CTPS1KDM1AGPR119MAPTRHOC
SCHEMBL6474127 0.92 CYSLTR2 (0.43) CTPS1MAPTTP53PPARALMNA
SCHEMBL6473587 0.91 TP53 (0.45) MAPTTP53PPARAPPARGLMNA
SCHEMBL6474643 0.90 CYSLTR2 (0.39) CTPS1KDM1AGPR119MAPTTP53
SCHEMBL6483737 0.89 SHMT2 (0.46) CTPS1MAPTTP53PPARAPPARG
SCHEMBL6474743 0.89 TP53 (0.44) MAPTTP53LMNA
SCHEMBL6479428 0.89 PPARA (0.41) CTPS1MAPTTP53PPARAPPARG
SCHEMBL6474952 0.88 PPARG (0.41) CTPS1MAPTTP53PPARGCYSLTR2
SCHEMBL9721963 0.85 CYSLTR2 (0.56) CTPS1KDM1AGPR119MAPTTP53
SCHEMBL6483863 0.84 PPARA (0.47) KDM1AMAPTPPARAPPARGCYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6930131-B2 Aryl substituted 3-ethoxy phenyl trifluoromethane sulfonamides for the treatment of non-insulin dependent diabetes mellitus (NIDDM) WYETH (US) 2005-08-16 US disclosed
US-20030203941-A1 Substituted phenyl compounds for the treatment of non-insulin dependent diabetes mellitus WYETH (US) 2003-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030203941-A1 Substituted phenyl compounds for the treatment of non-insulin dependent diabetes mellitus GPR119, INSR, SLC5A1 CTPS1 1446/4885KDM1A 1124/4885GPR119 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.