SCHEMBL6475724

SCHEMBL6475724

O=S(=O)(Nc1cccc(CCOCc2csc(-c3ccc(F)c(Cl)c3)n2)c1)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.42
CTPS1 P17812 1/20 0.42
POLB P06746 2/20 0.40
MAPT P10636 4/20 0.37
CYSLTR2 Q9NS75 1/20 0.37
CYSLTR1 Q9Y271 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
PPARA Q07869 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 2/20 0.36
KDM1A O60341 1/20 0.36
RHOC P08134 1/20 0.35
RHOA P61586 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6482379 0.92 CTPS1 (0.43) TP53CTPS1MAPTCYSLTR2CYSLTR1
SCHEMBL6474127 0.88 CYSLTR2 (0.43) TP53CTPS1MAPTCYSLTR2CYSLTR1
SCHEMBL6473587 0.87 TP53 (0.45) TP53POLBMAPTPPARASMN1; SMN2
SCHEMBL6474643 0.86 CYSLTR2 (0.39) TP53CTPS1POLBMAPTCYSLTR2
SCHEMBL6474952 0.86 PPARG (0.41) TP53CTPS1MAPTCYSLTR2CYSLTR1
SCHEMBL6474743 0.85 TP53 (0.44) TP53MAPTRXFP1SMN1; SMN2LMNA
SCHEMBL6483737 0.85 SHMT2 (0.46) TP53CTPS1MAPTCYSLTR2CYSLTR1
SCHEMBL6479428 0.85 PPARA (0.41) TP53CTPS1POLBMAPTCYSLTR2
SCHEMBL6477943 0.80 CYSLTR2 (0.41) TP53CTPS1POLBCYSLTR2CYSLTR1
SCHEMBL6474761 0.78 CYSLTR2 (0.39) TP53CTPS1POLBMAPTCYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6930131-B2 Aryl substituted 3-ethoxy phenyl trifluoromethane sulfonamides for the treatment of non-insulin dependent diabetes mellitus (NIDDM) WYETH (US) 2005-08-16 US disclosed
US-20030203941-A1 Substituted phenyl compounds for the treatment of non-insulin dependent diabetes mellitus WYETH (US) 2003-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030203941-A1 Substituted phenyl compounds for the treatment of non-insulin dependent diabetes mellitus GPR119, INSR, SLC5A1 TP53 3797/4885CTPS1 1446/4885POLB 3924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.