SCHEMBL6486173

SCHEMBL6486173

CC(C)(C)NC(=O)c1ncccn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.54
SMN1; SMN2 Q16637 5/20 0.47
RIPK1 Q13546 1/20 0.43
ALDH1A1 P00352 3/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 1/20 0.41
ANO1 Q5XXA6 1/20 0.40
NPC1 O15118 2/20 0.39
GAA P10253 2/20 0.39
RAB9A P51151 2/20 0.39
POLB P06746 2/20 0.39
HPGD P15428 2/20 0.39
CYP2C9 P11712 1/20 0.38
APEX1 P27695 1/20 0.38
EPHX1 P07099 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6415380 0.80 CNR2 (0.52) P2RX7NPC1RAB9ACYP2C9KMT2A
SCHEMBL16653076 0.78 P2RX7 (0.54) P2RX7SMN1; SMN2LMNATSHRNPC1
SCHEMBL13388574 0.78 HPGDS (0.36) SMN1; SMN2RIPK1ALDH1A1LMNAL3MBTL1
SCHEMBL2538917 0.78 NPC1 (0.41) SMN1; SMN2ALDH1A1LMNAL3MBTL1NPC1
SCHEMBL161652 0.77 SMN1; SMN2 (0.39) SMN1; SMN2RIPK1ALDH1A1LMNAL3MBTL1
SCHEMBL1834472 0.76 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1LMNAL3MBTL1NPC1
SCHEMBL2363536 0.75 P2RX7 (0.60) P2RX7RIPK1ALDH1A1LMNANPC1
SCHEMBL26750121 0.74 P2RX7 (0.53) P2RX7TSHR
SCHEMBL163050 0.74 SMN1; SMN2 (0.58) P2RX7SMN1; SMN2RIPK1ALDH1A1TSHR
SCHEMBL268817 0.74 P2RX7 (0.65) P2RX7SMN1; SMN2RIPK1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103582629-B As 5-(phenyl/pyridyl-ethynyl)-2-pyridine/2-pyrimidine-methane amide of MGLUR5 conditioning agent HOFFMAN-LA ROCHE LTD. (CH) 2015-10-07 CN claimed
CN-113072489-A Preparation method of nitrogen heteroaromatic ring formamide compound 湖北工业大学 2021-07-06 CN disclosed
CN-103582629-B As 5-(phenyl/pyridyl-ethynyl)-2-pyridine/2-pyrimidine-methane amide of MGLUR5 conditioning agent HOFFMAN-LA ROCHE LTD. (CH) 2015-10-07 CN disclosed
US-6939872-B2 2-anilino-pyrimidine derivatives as cyclin dependent kinase inhibitors ASTRAZENECA AB (SE) 2005-09-06 US disclosed