SCHEMBL6489284

SCHEMBL6489284

Cc1cc(CNc2cccc(C(=O)O)c2)cc2c1nc(C)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 8/20 0.50
MRGPRX4 Q96LA9 2/20 0.42
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PPARG P37231 1/20 0.40
DCTPP1 Q9H773 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGDR Q13258 1/20 0.39
CCR2 P41597 1/20 0.39
PIK3C2B O00750 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6487974 0.90 MAPT (0.42) PPARAMAPTMEN1KMT2ANPSR1
SCHEMBL6501562 0.84 NR4A2 (0.57) MRGPRX4PPARG
SCHEMBL6491218 0.83 CD38 (0.44) NPSR1PPARGDCTPP1ALDH1A1L3MBTL1
SCHEMBL6488659 0.82 PPARA (0.43) PPARAMRGPRX4NPSR1PPARGDCTPP1
SCHEMBL6490645 0.82 PTGDR (0.44) MRGPRX4NPSR1PPARGDCTPP1L3MBTL1
SCHEMBL6172911 0.81 PPARG (0.48) MRGPRX4NPSR1PPARGDCTPP1ALDH1A1
SCHEMBL6489657 0.79 KDM4C (0.42) MRGPRX4PPARGDCTPP1
SCHEMBL6489915 0.78 NR4A2 (0.46) MRGPRX4MAPTPPARGDCTPP1
SCHEMBL6500955 0.78 KDM4C (0.40) MRGPRX4PPARGDCTPP1PIK3C2B
SCHEMBL7200058 0.78 FABP3 (0.48) MRGPRX4PIK3C2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050014812-A1 Benzimidazole compounds FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-01-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014812-A1 Benzimidazole compounds SLC5A1, SLC5A2, G6PD PPARA 665/4885MRGPRX4 2443/4885MAPT 3168/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.