SCHEMBL6490645

SCHEMBL6490645

Cc1cc(-c2cccc(C(=O)O)c2)cc2c1nc(C)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 1/20 0.44
EIF4EBP1 Q13541 3/20 0.42
NR4A1 P22736 1/20 0.42
NR4A2 P43354 1/20 0.42
NR4A3 Q92570 1/20 0.42
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
ALOX5AP P20292 1/20 0.42
PPARG P37231 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
DCTPP1 Q9H773 1/20 0.41
PIK3C2B O00750 2/20 0.41
MRGPRX4 Q96LA9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6496733 0.92 ALOX5AP (0.47) RXRARXRBALOX5APPPARGTSHR
SCHEMBL6489563 0.90 SMN1; SMN2 (0.52) RXRARXRBALOX5APPPARGTSHR
SCHEMBL6488966 0.87 RXRA (0.41) EIF4EBP1NR4A1NR4A2NR4A3RXRA
SCHEMBL6494714 0.87 KDM4C (0.44) PTGDRNR4A1NR4A2NR4A3PPARG
SCHEMBL6487982 0.86 DCTPP1 (0.41) EIF4EBP1RXRARXRBALOX5APPPARG
SCHEMBL6491734 0.86 PPARG (0.53) PTGDREIF4EBP1NR4A1NR4A2NR4A3
SCHEMBL6498703 0.86 LMNA (0.39) PPARGNPSR1CYP1A2CYP3A4CYP2D6
SCHEMBL6172911 0.86 PPARG (0.48) NR4A2PPARGNPSR1CYP1A2CYP3A4
SCHEMBL6497678 0.85 PTPN11 (0.46) EIF4EBP1PPARG
SCHEMBL6487328 0.85 RXRA (0.40) EIF4EBP1RXRARXRBPPARGDCTPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050014812-A1 Benzimidazole compounds FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-01-20 US disclosed
WO-2004108686-A2 BENZIMIDAZOLE COMPOUNDS HAVING HYPOGLYCEMIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014812-A1 Benzimidazole compounds SLC5A1, SLC5A2, G6PD PTGDR 3383/4885EIF4EBP1 1623/4885NR4A1 1583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.