SCHEMBL6498161

SCHEMBL6498161

c1ccc(CN2CCCC3(CCN(Cc4cccc(Oc5ccccc5)c4)CC3)C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.60
ALDH1A1 P00352 4/20 0.60
CYP3A4 P08684 4/20 0.60
TSHR P16473 4/20 0.60
CCR8 P51685 3/20 0.58
KCNH2 Q12809 3/20 0.58
KDM4E B2RXH2 2/20 0.57
TDP1 Q9NUW8 1/20 0.57
HPGD P15428 1/20 0.57
HTT P42858 1/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
FAAH O00519 2/20 0.54
MGLL Q99685 1/20 0.53
TRPV6 Q9H1D0 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499571 0.83 ALDH1A1 (0.75) ALDH1A1CCR8KDM4ETDP1HPGD
SCHEMBL6496864 0.81 ALDH1A1 (0.73) ALDH1A1CCR8KDM4ETDP1HPGD
SCHEMBL13743319 0.80 ALDH1A1 (0.70) CYP2D6ALDH1A1TSHRCCR8KCNH2
SCHEMBL6506121 0.79 CCR8 (0.57) ALDH1A1CCR8KCNH2KDM4ETDP1
Hydrochloric Acid SCHEMBL4186299 0.79 ALDH1A1 (0.68) CYP2D6ALDH1A1TSHRCCR8KCNH2
SCHEMBL2791333 0.79 FAAH (0.71) CCR8KCNH2FAAHMGLL
SCHEMBL24798927 0.78 CYP2D6 (0.68) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL24798656 0.78 CYP2D6 (0.68) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
Hydrochloric Acid SCHEMBL896900 0.78 FAAH (0.58) CYP2D6ALDH1A1CCR8KCNH2FAAH
SCHEMBL5197063 0.78 CCR8 (0.74) CYP2D6ALDH1A1CYP3A4CCR8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050143372-A1 Compounds, pharmaceutical compositions and methods of use therefor MILLENNIUM PHARMACEUTICALS, INC. 2005-06-30 US disclosed
WO-2003037271-A2 COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREFOR MILLENNIUM PHARMACEUTICALS,INC. (US) 2003-05-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143372-A1 Compounds, pharmaceutical compositions and methods of use therefor CCR8, CCL11, CCR5 CYP2D6 1424/4885ALDH1A1 1071/4885CYP3A4 1514/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.