SCHEMBL6499280

SCHEMBL6499280

O=C(O)CC(Cc1ccc(O)cc1)c1nc(C(F)(F)F)cs1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.39
ESR1 P03372 5/20 0.37
ESR2 Q92731 5/20 0.37
ACE P12821 1/20 0.36
SLC7A5 Q01650 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
FFAR1 O14842 1/20 0.34
MIF P14174 1/20 0.34
GCGR P47871 1/20 0.33
GIPR P48546 1/20 0.33
CA2 P00918 1/20 0.33
CAMK2A Q9UQM7 1/20 0.33
PTPRB P23467 2/20 0.33
PTGER1 P34995 1/20 0.33
PTGS2 P35354 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32
NAALAD2 Q9Y3Q0 1/20 0.32
PTGES O14684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7803616 0.86 ESR1 (0.37) PKMESR1ESR2ACEMIF
SCHEMBL6501114 0.85 FFAR1 (0.49) PKMFFAR1ITGB3ITGAV
SCHEMBL8370944 0.84 ESR1 (0.48) ESR1ESR2PTPRBPTGS2PTGES
SCHEMBL6176693 0.81 PKM (0.44) PKMESR1ESR2SLC7A5FFAR1
SCHEMBL6500369 0.81 AKR1B1 (0.37) PKMPTPRBPTGER1
SCHEMBL1822558 0.75 ITGB3 (0.69) ITGB3ITGAV
SCHEMBL6175673 0.73 CTSA (0.45) PKMSLC7A5
SCHEMBL6179589 0.73 CTSA (0.45) PKMSLC7A5
SCHEMBL6177067 0.73 CTSA (0.45) PKMSLC7A5
SCHEMBL6490172 0.71 ESR1 (0.49) ESR1ESR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6881736-B1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2005-04-19 US disclosed
EP-1218005-B1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-12-15 EP disclosed
EP-1218005-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-10-09 EP disclosed
EP-1218005-A2 VITRONECTIN RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-07-03 EP disclosed
WO-2001017959-A2 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-03-15 WO disclosed