SCHEMBL6500369

SCHEMBL6500369

O=C(O)CC(Cc1ccccc1O)c1nc(C(F)(F)F)cs1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.37
PTPRB P23467 2/20 0.35
IDH2 P48735 1/20 0.34
PKM P14618 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
ROCK1 Q13464 1/20 0.33
EEF2K O00418 1/20 0.33
POLB P06746 2/20 0.32
GAA P10253 1/20 0.32
KCNH2 Q12809 2/20 0.32
LMNA P02545 1/20 0.32
GABBR2 O75899 1/20 0.31
GABBR1 Q9UBS5 1/20 0.31
PTGER1 P34995 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499280 0.81 PKM (0.39) PTPRBPKMPTGER1
SCHEMBL6501114 0.76 FFAR1 (0.49) PKM
SCHEMBL6179146 0.71 GABBR2 (0.56) AKR1B1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL6179138 0.71 GABBR2 (0.56) AKR1B1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL7803616 0.68 ESR1 (0.37) PTPRBPKMMEN1KMT2A
SCHEMBL6493607 0.65 ITGB3 (0.47) AKR1B1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6493595 0.65 ITGB3 (0.47) AKR1B1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8370944 0.64 ESR1 (0.48) PTPRBSLC6A2
SCHEMBL9863542 0.63 AKR1B1 (0.55) AKR1B1MAPK1POLBALDH1A1
SCHEMBL20876112 0.63 CPA1 (0.62) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6881736-B1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2005-04-19 US disclosed