SCHEMBL6501406

SCHEMBL6501406

CC(C)(C)OC(=O)Nc1cc(-c2cccc(Nc3ccccc3)c2)ccn1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIP5K1C O60331 9/20 0.54
PIK3CA P42336 9/20 0.54
MAPK8 P45983 8/20 0.53
MAPK10 P53779 8/20 0.53
CYP17A1 P05093 1/20 0.50
ACVRL1 P37023 1/20 0.49
PIP5K1B O14986 3/20 0.48
PIP5K1A Q99755 3/20 0.48
PIK3CD O00329 2/20 0.48
PDGFRB P09619 2/20 0.48
PIK3CB P42338 2/20 0.48
PI4KA P42356 2/20 0.48
PIK3CG P48736 2/20 0.48
PDK1 Q15118 2/20 0.48
PI4KB Q9UBF8 2/20 0.48
MAPK14 Q16539 2/20 0.48
EGFR P00533 1/20 0.47
CNR1 P21554 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5251219 0.90 EGFR (0.57) MAPK8MAPK10CYP17A1EGFRCNR1
SCHEMBL6507767 0.87 PIP5K1C (0.58) PIP5K1CPIK3CAMAPK8MAPK10PIP5K1B
SCHEMBL6502882 0.83 IRAK4 (0.49) CYP17A1EGFR
SCHEMBL6507708 0.82 PIP5K1C (0.63) PIP5K1CPIK3CAMAPK8MAPK10ACVRL1
SCHEMBL24010535 0.81 BRAF (0.57)
SCHEMBL1518666 0.80 MAPK10 (0.70) PIP5K1CPIK3CAMAPK8MAPK10ACVRL1
SCHEMBL24004071 0.80 ACVRL1 (0.47) CYP17A1ACVRL1
SCHEMBL13754832 0.79 CYP17A1 (0.64) CYP17A1
SCHEMBL5544966 0.79 CYP17A1 (0.47) CYP17A1EGFR
SCHEMBL8670718 0.79 FDPS (0.50) CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003123-A1 NOVEL PYRIDINE DERIVATIVES AS JNK SPECIFIC INHIBITORS ASTRAZENECA AB (SE) 2005-01-13 WO disclosed