SCHEMBL65021

SCHEMBL65021

COc1ccccc1CO[C]=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.58
TAAR1 Q96RJ0 1/20 0.48
ABCB1 P08183 1/20 0.47
CHRM2 P08172 3/20 0.47
CHRM1 P11229 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
HTT P42858 2/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
ATM Q13315 1/20 0.45
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
CA4 P22748 1/20 0.44
CA7 P43166 1/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1807876 0.84 ABCB1 (0.50) ABCB1L3MBTL1ALDH1A1GAACA12
SCHEMBL7531320 0.82 KMT2A (0.43) IDO1TAAR1CHRM2CHRM1L3MBTL1
SCHEMBL1054893 0.81 L3MBTL1 (0.56) L3MBTL1ALDH1A1GAAMAPTATM
SCHEMBL2088631 0.80 FFAR4 (0.43) IDO1ALDH1A1MAPTHPGDKDM4E
SCHEMBL11324512 0.80 ABCB1 (0.62) ABCB1L3MBTL1MAPTATMHPGD
SCHEMBL1129749 0.79 PTGS2 (0.46) ALDH1A1MAPTHPGDKDM4E
SCHEMBL8698021 0.79 L3MBTL1 (0.49) L3MBTL1ALDH1A1MAPTATMHPGD
SCHEMBL2096467 0.78 CA1 (0.41) IDO1ALDH1A1MAPTCA12CA1
SCHEMBL7644217 0.78 HRH1 (0.51) GAA
SCHEMBL5984175 0.78 GABRA1 (0.41) IDO1L3MBTL1MAPTATMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1991 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111187281-A Cephalosporin derivative containing guanidyl and preparation method thereof 广西科技大学 2020-05-22 CN claimed
EP-2976092-B1 CHEMICAL CROSSLINKERS AMICUS THERAPEUTICS INC (US) 2020-04-22 EP claimed
EP-3532475-A2 PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF Array Biopharma Inc. (US) 2019-09-04 EP claimed
WO-2019005796-A1 PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF ZHAO QIAN (US) 2019-01-03 WO claimed
WO-2018081417-A2 PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF ZHAO QIAN (US) 2018-05-03 WO claimed
CN-107530259-A Method using acid amides, acid or ester C glycosides derivatives processing keratin material and the cosmetic composition containing them 莱雅公司 2018-01-02 CN claimed
CN-104829632-B A kind of cephalosporins derivatives of the substituent containing aminodithioformic acid 中山大学 2017-09-29 CN claimed
CN-104530417-B A kind of multiple functionalized H types polyethyleneglycol derivative and preparation method thereof 厦门赛诺邦格生物科技股份有限公司 2017-09-08 CN claimed
CN-104530415-B A kind of different functionalization Y types polyethyleneglycol derivative, preparation method and its bio-related substance 厦门赛诺邦格生物科技股份有限公司 2017-09-01 CN claimed
EP-3068770-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINYLCYCLOPENTANE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2016-09-21 EP claimed
WO-1995006030-A1 HYDROXYETHYLAMINO SULPHONAMIDES USEFUL AS RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1995-03-02 WO claimed
US-5393878-A Pyrimidine nucleosides having cyclopentafuran skeleton CIBA-GEIGY CORPORATION (US) 1995-02-28 US claimed
WO-1994018329-A2 SERINE PROTEASE VARIANTS HAVING PEPTIDE LIGASE ACTIVITY GENENTECH, INC. (US) 1994-08-18 WO claimed
US-5319080-A Antiviral agents CIBA-GEIGY CORPORATION (US) 1994-06-07 US claimed
EP-0583338-A1 METHOD FOR SYNTHESIZING PEPTIDES, NOVEL AMINO ACID DERIVATIVES USED THEREIN, AND METHODS FOR PREPARING SAME. PROPEPTIDE SA (FR) 1994-02-23 EP claimed
WO-1992019643-A1 METHOD FOR SYNTHESIZING PEPTIDES, NOVEL AMINO ACID DERIVATIVES USED THEREIN, AND METHODS FOR PREPARING SAME PROPEPTIDE (FR) 1992-11-12 WO claimed
EP-0268963-A1 Benzazolylthio-carbapenem antibiotics BAYER AG (DE) 1988-06-01 EP claimed
EP-0053962-B1 CEPHALOSPORIN DERIVATIVES AND THEIR PREPARATION RHONE-POULENC SANTE (FR) 1985-03-13 EP claimed
US-4393228-A THIOL PROTEASE INHIBITORS, ANTIINFLAMMATORY TAISHO PHARMACEUTICAL CO., LTD. (JP) 1983-07-12 US claimed
US-4180571-A Arylmalonamido-1-oxadethiacephalosporins SHIONOGI & CO., LTD. (JP) 1979-12-25 US claimed