SCHEMBL6502342

SCHEMBL6502342

CC(C)(C)COC(=O)N[C@@H](Cc1ccc2c(c1)C(=O)CC(O)(CCCN(C(=O)OCC(Cl)(Cl)Cl)c1ccccn1)O2)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.36
ITGAV P06756 1/20 0.36
ITGA4 P13612 4/20 0.32
ITGB1 P05556 3/20 0.32
ITGA2B P08514 2/20 0.31
ITGB7 P26010 1/20 0.31
MEN1 O00255 1/20 0.30
GMNN O75496 1/20 0.30
EGFR P00533 1/20 0.30
LMNA P02545 1/20 0.30
CYP3A4 P08684 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
ADRB3 P13945 1/20 0.30
TSHR P16473 1/20 0.30
ADRA2B P18089 1/20 0.30
NFKB1 P19838 1/20 0.30
TACR2 P21452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6493594 0.80 ITGB3 (0.43) ITGB3ITGAVITGA4ITGB1ITGA2B
SCHEMBL6493907 0.79 ITGB3 (0.42) ITGB3ITGAVITGA4ITGB1ITGA2B
SCHEMBL6503598 0.77 ITGB1 (0.37) ITGB3ITGAVITGA4ITGB1ITGA2B
SCHEMBL5204549 0.73 ITGB3 (0.37) ITGB3ITGAVITGA2BMEN1CYP3A4
SCHEMBL5202520 0.73 ITGB3 (0.37) ITGB3ITGAVKMT2AHSD17B10
SCHEMBL5207840 0.71 MAPT (0.32) ITGB3ITGAVITGB1LMNAMAPT
SCHEMBL14431254 0.71 MAPT (0.32) ITGB3ITGAVITGB1LMNAMAPT
SCHEMBL6494232 0.67 MAPT (0.30) MAPT
SCHEMBL6495275 0.66 ITGB3 (0.36) ITGB3ITGAVITGA4ITGB1ITGA2B
SCHEMBL6495566 0.63 FFAR1 (0.43) LMNACYP3A4CYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849646-B1 Chromenone and chromanone derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2005-02-01 US disclosed