SCHEMBL6503598

SCHEMBL6503598

CC(C)(C)COC(=O)N[C@@H](Cc1ccc2oc(CCCN(C(=O)OCC(Cl)(Cl)Cl)c3ccccn3)cc(=O)c2c1)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.37
ITGA5 P08648 1/20 0.37
ITGB3 P05106 4/20 0.36
ITGAV P06756 1/20 0.36
TYR P14679 1/20 0.34
ITGA2B P08514 3/20 0.33
MAPT P10636 2/20 0.33
PPARG P37231 4/20 0.32
PPARA Q07869 3/20 0.32
ITGA4 P13612 1/20 0.31
ITGB7 P26010 1/20 0.31
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
PRSS3 P35030 1/20 0.31
TPSAB1 Q15661 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
CAPN1 P07384 1/20 0.30
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14431254 0.94 MAPT (0.32) ITGB1ITGA5ITGB3ITGAVTYR
SCHEMBL5207840 0.94 MAPT (0.32) ITGB1ITGA5ITGB3ITGAVTYR
SCHEMBL6495275 0.89 ITGB3 (0.36) ITGB1ITGA5ITGB3ITGAVTYR
SCHEMBL5203778 0.83 ITGB3 (0.32) ITGB3ITGAV
SCHEMBL14431255 0.81 ITGB1 (0.50) ITGB1ITGA5ITGB3ITGAVTYR
SCHEMBL3048694 0.81 ITGB1 (0.50) ITGB1ITGA5ITGB3ITGAVTYR
SCHEMBL6498071 0.79 ITGB3 (0.44) ITGB3ITGAVTYRITGA2BPPARG
SCHEMBL3052420 0.79 ITGB3 (0.44) ITGB3ITGAVTYRITGA2BPPARG
SCHEMBL6502618 0.78 TYR (0.44) ITGB3ITGAVTYRITGA2BPPARG
SCHEMBL6502342 0.77 ITGB3 (0.36) ITGB1ITGB3ITGAVITGA2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849646-B1 Chromenone and chromanone derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2005-02-01 US disclosed