SCHEMBL5204549

SCHEMBL5204549

CCOC(=O)[C@H](Cc1ccc2c(c1)C(=O)CC(O)(CCCOCc1ccccc1)O2)NC(=O)OCC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.37
ITGAV P06756 3/20 0.37
TYR P14679 1/20 0.35
ITGA2B P08514 4/20 0.35
PPARA Q07869 1/20 0.34
TSHR P16473 3/20 0.33
TACR1 P25103 1/20 0.33
CTSK P43235 1/20 0.33
CYP3A4 P08684 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6493907 0.94 ITGB3 (0.42) ITGB3ITGAVTYRITGA2BPPARA
SCHEMBL5202520 0.90 ITGB3 (0.37) ITGB3ITGAVTACR1CTSKALDH1A1
SCHEMBL6493594 0.84 ITGB3 (0.43) ITGB3ITGAVTYRITGA2BALDH1A1
SCHEMBL5210309 0.74 TYR (0.41) ITGB3ITGAVTYRITGA2BPPARA
SCHEMBL6502342 0.73 ITGB3 (0.36) ITGB3ITGAVITGA2BPPARATSHR
SCHEMBL27406870 0.68 CTSL (0.48) ITGB3ITGAVTYRTSHRTACR1
SCHEMBL7361913 0.68 ALOX15 (0.40) ITGB3ITGAVITGA2BCTSK
SCHEMBL6440663 0.65 CTSL (0.64) TYRTACR1CTSKALDH1A1
SCHEMBL6440666 0.65 CTSL (0.64) TYRTACR1CTSKALDH1A1
SCHEMBL4679583 0.64 USP2 (0.39) ITGB3ITGAVTSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124824-B1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2007-08-22 EP disclosed