SCHEMBL6503228

SCHEMBL6503228

COc1ccc(CC(OC(C)C)C(=O)O)cc1C(C)NC(=O)c1cc(C)nn1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.45
SMYD3 Q9H7B4 1/20 0.45
TSHR P16473 1/20 0.43
KMT2A Q03164 6/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 1/20 0.40
MDM2 Q00987 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6494362 0.86 NPY5R (0.43)
SCHEMBL6503221 0.83 MAPT (0.54) ALDH1A1MAPTTSHRKMT2AL3MBTL1
SCHEMBL6502018 0.81 PHGDH (0.55)
SCHEMBL6505823 0.81 KMT2A (0.41) KMT2A
SCHEMBL6495617 0.78 MME (0.50)
SCHEMBL6505350 0.77 PPARG (0.40)
SCHEMBL6497349 0.77 OPRK1 (0.40) L3MBTL1
SCHEMBL6496485 0.77 HSD17B10 (0.52) ALDH1A1MAPTTSHRKMT2AMEN1
SCHEMBL6503168 0.76 KMT2A (0.39) KMT2AMEN1
SCHEMBL6504374 0.73 OPRK1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed