SCHEMBL6505484

SCHEMBL6505484

COC(=O)c1cc(C(N)=O)c(NC(N)=O)s1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.55
IKBKB O14920 9/20 0.51
JAK2 O60674 2/20 0.50
JAK3 P52333 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
EIF2AK2 P19525 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6505865 0.85 IKBKB (0.58) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6507152 0.84 IKBKB (0.57) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6514837 0.81 CHEK1 (0.47) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6507636 0.79 IKBKB (0.51) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL11921318 0.76 IKBKB (0.59) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6506816 0.76 CHEK1 (0.36) CHEK1IKBKBALDH1A1
SCHEMBL6511724 0.75 MAPT (0.51) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL1563630 0.74 CHEK1 (0.45) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6505745 0.74 IKBKB (0.57) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6510409 0.73 CHEK1 (0.44) CHEK1IKBKBJAK2JAK3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed