SCHEMBL6506816

SCHEMBL6506816

COC(=O)c1cc(NC=O)c(NC(N)=O)s1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 6/20 0.36
HPGD P15428 4/20 0.35
MAPK1 P28482 3/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
IKBKB O14920 3/20 0.34
CSNK2A2 P19784 1/20 0.34
KDR P35968 1/20 0.34
CSNK2B P67870 1/20 0.34
CSNK2A1 P68400 1/20 0.34
OPRD1 P41143 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
TSHR P16473 1/20 0.33
ATM Q13315 1/20 0.33
LMNA P02545 2/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6514944 0.87 KDM5A (0.37) CHEK1KDM4EALDH1A1IKBKBMAPT
SCHEMBL6506529 0.77 KDM5A (0.36) CHEK1IKBKB
SCHEMBL6512268 0.77 IKBKB (0.35) CHEK1MAPK1IKBKB
SCHEMBL6505484 0.76 CHEK1 (0.55) CHEK1ALDH1A1IKBKB
SCHEMBL6505649 0.74 IKBKB (0.45) CHEK1IKBKB
SCHEMBL6508772 0.73 IKBKB (0.38) CHEK1KDM4EIKBKB
SCHEMBL28374051 0.68 HDAC3 (0.47) HPGDMAPK1KDM4EALDH1A1CSNK2A2
SCHEMBL29749792 0.68 HDAC3 (0.47) HPGDMAPK1KDM4EALDH1A1CSNK2A2
SCHEMBL6509499 0.66 PTK2 (0.40) MAPK1ALDH1A1MAPT
SCHEMBL9722819 0.66 ALDH1A1 (0.45) HPGDMAPK1KDM4EALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed