SCHEMBL6506047

SCHEMBL6506047

CC(Oc1ccc(F)cc1)c1cccc(N2CCC(C(=O)O)CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 6/20 0.57
S1PR5 Q9H228 2/20 0.46
S1PR1 P21453 1/20 0.46
SCN9A Q15858 2/20 0.46
ACACB O00763 1/20 0.43
FFAR4 Q5NUL3 1/20 0.42
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6507338 0.87 LGMN (0.49) NOTUM
SCHEMBL6502769 0.80 SCN9A (0.59) NOTUMSCN9AFFAR4PPARA
SCHEMBL31381267 0.80 NOTUM (0.67) NOTUMACACB
SCHEMBL6506958 0.80 NOTUM (0.85) NOTUM
SCHEMBL5799166 0.76 NOTUM (0.58) NOTUM
SCHEMBL6499932 0.76 CYP4F2 (0.61) NOTUMS1PR5S1PR1
SCHEMBL15578214 0.75 HTR1A (0.58) NOTUMS1PR1SCN9AFFAR4
SCHEMBL5798727 0.73 NOTUM (0.59) NOTUMFFAR4
SCHEMBL23381187 0.73 NOTUM (1.00) NOTUM
SCHEMBL1749207 0.72 NOTUM (0.81) NOTUMSCN9AFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed