SCHEMBL6506181

SCHEMBL6506181

O=[N+]([O-])c1[c]cc(Br)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MAPT P10636 3/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 2/20 0.34
VCP P55072 1/20 0.34
ALDH1A1 P00352 3/20 0.32
HIF1A Q16665 1/20 0.32
CYP3A4 P08684 1/20 0.32
VCAM1 P19320 1/20 0.31
GLA P06280 1/20 0.31
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11909458 0.85 VCP (0.38) ATMTDP1MAPTPKMMAPK1
SCHEMBL4577560 0.82 ATM (0.36) ATMTDP1ALDH1A1HIF1AVCAM1
SCHEMBL28774035 0.77 ALDH1A1 (0.36) ATMTDP1MAPTMAPK1ALDH1A1
SCHEMBL27818989 0.77 ALDH1A1 (0.33) TDP1ALDH1A1HIF1ACYP3A4
SCHEMBL1822058 0.74 ALDH1A1 (0.46) ATMTDP1MAPTPKMMAPK1
SCHEMBL27684781 0.73 ALDH1A1 (0.36) ATMTDP1MAPTMAPK1ALDH1A1
SCHEMBL4902091 0.73 CA12 (0.34) TDP1MAPTMAPK1ALDH1A1HIF1A
SCHEMBL28738082 0.73 HTT (0.38) TDP1MAPTPKMALDH1A1CYP3A4
SCHEMBL9304210 0.70 ALDH1A1 (0.33) ATMTDP1MAPTMAPK1ALDH1A1
SCHEMBL3279026 0.69 GRIN2D (0.37) MAPTMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO claimed
CN-112867721-B STING agonistic compounds 小野药品工业株式会社 2023-12-08 CN disclosed
CN-112867721-A STING agonistic compounds 小野药品工业株式会社 2021-05-28 CN disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed