SCHEMBL6506646

SCHEMBL6506646

COC(=O)[C@H](CN1CCCC1=O)NC(=O)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 4/20 0.59
KYNU Q16719 1/20 0.51
LMNA P02545 1/20 0.49
ALDH1A1 P00352 1/20 0.49
ALOX15 P16050 1/20 0.49
OPRK1 P41145 1/20 0.48
CTSK P43235 7/20 0.47
CTSL P07711 4/20 0.47
CTSB P07858 3/20 0.47
CTSS P25774 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8142600 0.97 CASP1 (0.56) CASP1KYNULMNAALDH1A1ALOX15
SCHEMBL10443427 0.91 CASP1 (0.61) CASP1LMNAOPRK1CTSKCTSL
SCHEMBL10443426 0.91 CASP1 (0.61) CASP1LMNAOPRK1CTSKCTSL
SCHEMBL8142582 0.88 CASP1 (0.58) CASP1OPRK1CTSKCTSLCTSB
SCHEMBL12023182 0.83 CASP1 (0.53) CASP1LMNAOPRK1CTSKCTSL
SCHEMBL29440261 0.82 KYNU (0.51) CASP1KYNUALDH1A1ALOX15OPRK1
SCHEMBL29062923 0.81 ALDH1A1 (0.50) CASP1KYNUALDH1A1ALOX15OPRK1
SCHEMBL29062922 0.81 ALDH1A1 (0.50) CASP1KYNUALDH1A1ALOX15OPRK1
SCHEMBL7413795 0.79 CASP1 (0.74) CASP1
SCHEMBL6497607 0.78 CASP1 (0.61) CASP1KYNUALDH1A1ALOX15CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed
EP-0350163-A2 Renin inhibitory peptides BEECHAM GROUP PLC (GB) 1990-01-10 EP disclosed