SCHEMBL6497607

SCHEMBL6497607

COC(=O)C(CN1Cc2ccccc2C1=O)NC(=O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.61
KYNU Q16719 1/20 0.49
CTSL P07711 10/20 0.48
CTSB P07858 6/20 0.48
ITGAV P06756 1/20 0.48
ALOX15 P16050 2/20 0.47
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KDM4E B2RXH2 1/20 0.47
TSHR P16473 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
CTSK P43235 5/20 0.46
CTSS P25774 3/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8296213 1.00 CASP1 (0.61) CASP1KYNUCTSLCTSBITGAV
SCHEMBL15372554 0.82 CASP1 (0.47) CASP1KYNUCTSLCTSBALOX15
SCHEMBL6474852 0.80 ITGB3 (0.55) CASP1
SCHEMBL7331730 0.79 CTSL (0.42) CASP1KYNUCTSLCTSBALOX15
SCHEMBL29440261 0.78 KYNU (0.51) CASP1KYNUCTSLCTSBALOX15
SCHEMBL6506646 0.78 CASP1 (0.59) CASP1KYNUCTSLCTSBALOX15
SCHEMBL8297568 0.78 NPC1 (0.50) ITGAVALOX15RAB9ANPC1KDM4E
SCHEMBL8142600 0.77 CASP1 (0.56) CASP1KYNUCTSLCTSBALOX15
SCHEMBL29062923 0.77 ALDH1A1 (0.50) CASP1KYNUCTSLCTSBALOX15
SCHEMBL29062922 0.77 ALDH1A1 (0.50) CASP1KYNUCTSLCTSBALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed