SCHEMBL6506696

SCHEMBL6506696

Cc1ccccc1-n1cc(NC(N)=O)c(C(N)=O)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 1/20 0.56
IRAK4 Q9NWZ3 7/20 0.40
KDM4E B2RXH2 2/20 0.40
NR3C2 P08235 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 2/20 0.40
ADORA3 P0DMS8 3/20 0.39
ADORA2A P29274 2/20 0.39
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
KAT2B Q92831 1/20 0.38
EPHB4 P54760 1/20 0.37
HIF1A Q16665 1/20 0.37
EPAS1 Q99814 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6500409 0.85 ITK (0.55) ITKIRAK4KDM4EHTTSMN1; SMN2
SCHEMBL6467613 0.83 ITK (0.49) ITKIRAK4KDM4EHTTSMN1; SMN2
SCHEMBL6497350 0.80 ITK (0.49) ITKIRAK4KDM4EHTTSMN1; SMN2
SCHEMBL6469794 0.79 LMNA (0.47) ITKKDM4EHTTSMN1; SMN2POLB
SCHEMBL6501912 0.78 ITK (0.52) ITKIRAK4
SCHEMBL6503646 0.77 ITK (0.51) ITKIRAK4KDM4ENR3C2SMN1; SMN2
SCHEMBL6470399 0.77 ITK (0.44) ITKIRAK4KDM4ENR3C2HTT
SCHEMBL6468046 0.76 ITK (0.43) ITKKDM4ENR3C2HTTPOLB
SCHEMBL6500141 0.76 ITK (0.44) ITKIRAK4POLBALDH1A1MAPT
SCHEMBL6502246 0.76 ITK (0.44) ITKIRAK4LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050197338-A1 Substituted pyrazole urea compounds for the treatment of inflammation PHARMACIA AND UPJOHN COMPANY LLC 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197338-A1 Substituted pyrazole urea compounds for the treatment of inflammation IL4, ARG2, CASP4 ITK 4236/4885IRAK4 27/4885KDM4E 2424/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.