SCHEMBL6506837

SCHEMBL6506837

O=C(O)C1CCN(c2cncc3ccccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 9/20 0.53
CYP11B1 P15538 9/20 0.53
CDK8 P49336 2/20 0.47
NOTUM Q6P988 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP2C19 P33261 1/20 0.47
NEK2 P51955 1/20 0.46
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP46A1 Q9Y6A2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26103034 0.84 CYP11B2 (0.49) CYP11B2CYP11B1CDK8NOTUMKDM4E
SCHEMBL26103321 0.84 CYP11B2 (0.49) CYP11B2CYP11B1CDK8NOTUMKDM4E
SCHEMBL5802241 0.84 KDM4E (0.48) NOTUMKDM4ECYP2C19NEK2CYP46A1
SCHEMBL6500699 0.81 MAPT (0.55) CYP11B2CYP11B1CDK8KDM4EMEN1
SCHEMBL5780030 0.78 CYP11B2 (0.48) CYP11B2CYP11B1CDK8CYP46A1
SCHEMBL1728859 0.78 CYP11B2 (0.48) CYP11B2CYP11B1CDK8
SCHEMBL239284 0.77 CYP11B1 (0.52) CYP11B2CYP11B1CDK8
SCHEMBL27856065 0.76 CYP11B1 (0.61) CYP11B2CYP11B1CDK8ALDH1A1LMNA
SCHEMBL5820284 0.76 KDM4E (0.48) NOTUMKDM4ECYP2C19NEK2CYP46A1
SCHEMBL31342013 0.76 CYP11B1 (0.72) CYP11B2CYP11B1CDK8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050080113-A1 Medicinal compositions TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-04-14 US disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080113-A1 Medicinal compositions TNF, TRAF6, MMP8 CYP11B2 2363/4885CYP11B1 2166/4885CDK8 1974/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.