SCHEMBL6507023

SCHEMBL6507023

CC1(C)CC(=C(c2ccc(O)cc2)c2ccc(-c3ccccc3)cc2/C=C/C(=O)O)CC(C)(C)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ESR2 Q92731 3/20 0.34
BCL2L1 Q07817 1/20 0.34
BAD Q92934 1/20 0.34
PGR P06401 1/20 0.34
RELA Q04206 1/20 0.34
ALOX5 P09917 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
NFKB1 P19838 1/20 0.33
CA4 P22748 1/20 0.33
IP6K1 Q92551 1/20 0.33
IP6K3 Q96PC2 1/20 0.33
IP6K2 Q9UHH9 1/20 0.33
MIF P14174 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3468323 0.83 RELA (0.50) ESR1MEN1KMT2AESR2PGR
SCHEMBL3468317 0.83 RELA (0.50) ESR1MEN1KMT2AESR2PGR
SCHEMBL3468563 0.78 MMP3 (0.47) ESR1MEN1KMT2AESR2BCL2L1
SCHEMBL3467807 0.77 ESR1 (0.55) ESR1MEN1KMT2AESR2PGR
SCHEMBL3467812 0.77 ESR1 (0.55) ESR1MEN1KMT2AESR2PGR
SCHEMBL3468706 0.76 KMO (0.47) ESR1MEN1KMT2ALMNAMAPT
SCHEMBL3468080 0.73 ESR1 (0.51) ESR1MEN1KMT2ABCL2L1BAD
SCHEMBL3075249 0.73 ESR1 (0.49) ESR1ESR2PGRMAPTCA1
SCHEMBL3075252 0.73 ESR1 (0.49) ESR1ESR2PGRMAPTCA1
SCHEMBL27640751 0.73 ESR1 (0.39) ESR1MEN1KMT2AESR2BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005012220-A9 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF ESTROGEN RECEPTOR SMITHKLINE BEECHAM CORP (US) 2005-05-19 WO disclosed